Signaling peptide receptor

Signaling peptide receptor is a type of receptor which binds one or more signaling peptides or signaling proteins.

An example is the tropomyosin receptor kinase B (TrkB), which is bound and activated by the neurotrophic protein brain-derived neurotrophic factor (BDNF). Another example is the μ-opioid receptor (MOR), which is bound and activated by the opioid peptide hormone β-endorphin.

AdipoR1

 * Agonists
 * Peptide
 * Adiponectin
 * ADP-355
 * ADP-399
 * Non-peptide
 * AdipoRon
 * (–)-Arctigenin
 * Arctiin
 * Gramine
 * Matairesinol
 * Antagonists
 * Peptide
 * ADP-400

AdipoR2

 * Agonists
 * Peptide
 * Adiponectin
 * ADP-355
 * ADP-399
 * Non-peptide
 * AdipoRon
 * Deoxyschizandrin
 * Parthenolide
 * Syringing
 * Taxifoliol
 * Antagonists
 * Peptide
 * ADP-400

Bradykinin receptor

 * Agonists
 * Bradykinin
 * Kallidin
 * Antagonists
 * FR-173657
 * Icatibant
 * LF22-0542

Calcitonin gene-related peptide receptor

 * Agonists
 * Amylin
 * CGRP
 * Pramlintide
 * Antagonists
 * Atogepant
 * BI 44370 TA
 * CGRP (8-37)
 * MK-3207
 * Olcegepant
 * Rimegepant
 * SB-268262
 * Telcagepant
 * Ubrogepant
 * Antibodies
 * Eptinezumab
 * Erenumab
 * Fremanezumab
 * Galcanezumab

CCKA

 * Agonists
 * Cholecystokinin
 * Antagonists
 * Amiglumide
 * Asperlicin
 * Devazepide
 * Dexloxiglumide
 * Lintitript
 * Lorglumide
 * Loxiglumide
 * Pranazepide
 * Proglumide
 * Tarazepide
 * Tomoglumide

CCKB

 * Agonists
 * Cholecystokinin
 * CCK-4
 * Gastrin
 * Pentagastrin (CCK-5)
 * Antagonists
 * Ceclazepide
 * CI-988 (PD-134308)
 * Itriglumide
 * L-365,360
 * Netazepide
 * Proglumide
 * Spiroglumide

Unsorted

 * Antagonists
 * Nastorazepide

CRF1

 * Agonists
 * Cortagine
 * Corticorelin
 * Corticotropin-releasing hormone
 * Sauvagine
 * Stressin I
 * Urocortin
 * Antagonists
 * Antalarmin
 * Astressin-B
 * CP-154,526
 * Emicerfont
 * Hypericin
 * LWH-234
 * NBI-27914
 * NBI-74788
 * Pexacerfont
 * R-121919
 * TS-041
 * Verucerfont

CRF2

 * Agonists
 * Corticorelin
 * Corticotropin-releasing hormone
 * Sauvagine
 * Urocortin
 * Antagonists
 * Astressin-B

Endothelin receptor

 * Agonists
 * Endothelin 1
 * Endothelin 2
 * Endothelin 3
 * IRL-1620
 * Sarafotoxin
 * Antagonists
 * A-192621
 * Ambrisentan
 * Aprocitentan
 * Atrasentan
 * Avosentan
 * Bosentan
 * BQ-123
 * BQ-788
 * Clazosentan
 * Darusentan
 * Edonentan
 * Enrasentan
 * Fandosentan
 * Feloprentan
 * Macitentan
 * Nebentan
 * Sitaxentan
 * Sparsentan
 * Tezosentan
 * Zibotentan

GAL1

 * Agonists
 * Galanin
 * Galanin (1-15)
 * Galanin-like peptide
 * Galmic
 * Galnon
 * NAX 810-2
 * Antagonists
 * C7
 * Dithiepine-1,1,4,4-tetroxide
 * Galantide (M15)
 * M32
 * M35
 * M40
 * SCH-202596

GAL2

 * Agonists
 * Galanin
 * Galanin (1-15)
 * Galanin (2-11)
 * Galanin-like peptide
 * Galmic
 * Galnon
 * J18
 * NAX 810-2
 * Antagonists
 * C7
 * Galantide (M15)
 * M32
 * M35
 * M40
 * M871

GAL3

 * Agonists
 * Galanin
 * Galanin (1-15)
 * Galmic
 * Galnon
 * Antagonists
 * C7
 * Galantide (M15)
 * GalR3ant
 * HT-2157
 * M32
 * M35
 * M40
 * SNAP-37889
 * SNAP-398299

GLP-1

 * Agonists
 * Albiglutide
 * Beinaglutide
 * Dulaglutide
 * Efpeglenatide
 * Exenatide
 * GLP-1
 * Langlenatide
 * Liraglutide
 * Lixisenatide
 * Oxyntomodulin
 * Pegapamodutide
 * Semaglutide
 * Taspoglutide

GLP-2

 * Agonists
 * Apraglutide
 * Elsiglutide
 * Glepaglutide
 * GLP-2
 * Teduglutide

Others

 * Propeptides
 * Preproglucagon
 * Proglucagon

Glucagon receptor

 * Agonists
 * Dasiglucagon
 * Glucagon
 * Oxyntomodulin
 * Antagonists
 * Adomeglivant
 * L-168,049
 * LGD-6972
 * Propeptides
 * Preproglucagon
 * Proglucagon

Insulin receptor

 * Agonists
 * Chaetochromin (4548-G05)
 * Insulin-like growth factor 1
 * Insulin-like growth factor 2
 * Insulin
 * Insulin aspart
 * Insulin degludec
 * Insulin detemir
 * Insulin glargine
 * Insulin glulisine
 * Insulin lispro
 * Mecasermin
 * Mecasermin rinfabate
 * Antagonists
 * BMS-754807
 * S661
 * S961
 * Kinase inhibitors
 * Linsitinib
 * Antibodies
 * Xentuzumab (against IGF-1 and IGF-2)

KiSS1-derived peptide receptor

 * Agonists
 * Kisspeptin (kisspeptin-54, metastin)
 * Kisspeptin-10
 * KISS1-305
 * MVT-602 (RVT-602, TAK-448)
 * TAK-683
 * Antagonists
 * Kisspeptin-234

Leptin receptor

 * Agonists
 * Leptin
 * Metreleptin

MCH1

 * Agonists
 * Melanin-concentrating hormone
 * Antagonists
 * ATC-0065
 * ATC-0175
 * GW-803430
 * NGD-4715
 * SNAP-7941
 * SNAP-94847

MCH2

 * Agonists
 * Melanin-concentrating hormone

Neuropeptide FF receptor

 * Agonists
 * Neuropeptide AF
 * Neuropeptide FF
 * Neuropeptide SF (RFRP-1)
 * Neuropeptide VF (RFRP-3)
 * Antagonists
 * BIBP-3226
 * RF9

Neuropeptide S receptor

 * Agonists
 * Neuropeptide S
 * Antagonists
 * ML-154
 * SHA-68

Y1

 * Agonists
 * Neuropeptide Y
 * Peptide YY
 * Antagonists
 * BIBO-3304
 * BIBP-3226
 * BVD-10
 * GR-231118
 * PD-160170

Y2

 * Agonists
 * 2-Thiouridine 5'-triphosphate
 * Neuropeptide Y
 * Neuropeptide Y (13-36)
 * Peptide YY
 * Peptide YY (3-36)
 * Antagonists
 * BIIE-0246
 * JNJ-5207787
 * SF-11

Y4

 * Agonists
 * GR-231118
 * Neuropeptide Y
 * Pancreatic polypeptide
 * Peptide YY
 * Antagonists
 * UR-AK49

Y5

 * Agonists
 * BWX-46
 * Neuropeptide Y
 * Peptide YY
 * Antagonists
 * CGP-71683
 * FMS-586
 * L-152,804
 * Lu AA-33810
 * MK-0557
 * NTNCB
 * Velneperit (S-2367)

NTS1

 * Agonists
 * Neurotensin
 * Neuromedin N
 * Antagonists
 * Meclinertant
 * SR-142948

NTS2

 * Agonists
 * Neurotensin
 * Antagonists
 * Levocabastine
 * SR-142948

Parathyroid hormone receptor

 * Agonists
 * Abaloparatide
 * Parathyroid hormone
 * Parathyroid hormone-related protein (PTHrP)
 * Semparatide
 * Teriparatide

Relaxin receptor

 * Agonists
 * Insulin-like factor 3
 * Relaxin (1, 2, 3)
 * Serelaxin

Thyrotropin-releasing hormone receptor

 * Agonists
 * Azetirelin
 * JTP-2942
 * Montirelin
 * Orotirelin
 * Posatirelin
 * Protirelin
 * Rovatirelin
 * RX-77368 (thymoliberin)
 * Taltirelin
 * TRH (TRF)

Thyrotropin receptor

 * Agonists
 * Thyrotropin alfa
 * TSH (thyrotropin)

VIPR1

 * Agonists
 * Peptide
 * Bay 55-9837
 * LBT-3393
 * PACAP
 * VIP

VIPR2

 * Agonists
 * Peptide
 * LBT-3627
 * PACAP
 * VIP

PAC1

 * Agonists
 * PACAP
 * PACAP (1-27)
 * PACAP (1-38)
 * Antagonists
 * PACAP (6-38)

Unsorted

 * PHI
 * PHM
 * PHV

Others

 * Endogenous
 * Adrenomedullin
 * Apelin
 * Asprosin
 * Bombesin
 * Calcitonin
 * Carnosine
 * CART
 * CLIP
 * DSIP
 * Enteroglucagon
 * Formyl peptide
 * GALP
 * GIP
 * GRP
 * Integrin ligands
 * collagens
 * fibrinogen
 * fibronectin
 * laminins
 * ICAM-1
 * ICAM-2
 * osteopontin
 * VCAM-1
 * vitronectin
 * Kininogens
 * Motilin
 * Natriuretic peptides
 * ANP
 * BNP
 * CNP
 * urodilatin
 * Nesfatin-1
 * Neuromedin B
 * Neuromedin N
 * Neuromedin S
 * Neuromedin U
 * Obestatin
 * Osteocalcin
 * Resistin
 * Secretin
 * Thymopoietin
 * Thymosins
 * Thymulin
 * Urotensin-II
 * VGF
 * Exogenous
 * Lifitegrast (LFA-1 antagonist)